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pro vyhledávání: '"Adeline Pretre"'
Autor:
Gordon Campbell, Anna Quattropani, Agnes Bombrun, Christophe Cleva, Marilène Gaudet, Gwenaelle Bouscary-Desforges, Marc Missotten, Stefano Crosignani, Hamina Daff, Kamel El Harkani, Tania Grippi-Vallotton, Nada Abla, Christèle Frémaux, Catherine Jorand-Lebrun, Zoë Johnson, Yves Humbert, Olivier Schott, Jean-François Arrighi, Charles G. Bradshaw, Mikaël Pâquet, Adeline Pretre, Pittet Pierre-Andre
Publikováno v:
ACS medicinal chemistry letters. 2(12)
Antagonism of the CRTH2 receptor represents a very attractive target for a variety of allergic diseases. Most CRTH2 antagonists known to date possess a carboxylic acid moiety, which is essential for binding. However, potential acid metabolites O-acyl