Zobrazeno 1 - 4
of 4
pro vyhledávání: '"Aaron Tieman"'
Autor:
Narayanan Hariharan, Kasim A. Mookhtiar, Liqun Gu, Jimmy Ren, Chen Sean, Ramakrishna Seethala, Michael Cap, Lori Kunselman, Min Zhou, Peter T. W. Cheng, William Fenderson, Chunning Shao, Cuixia Chu, Scott A. Biller, Hao Zhang, Fucheng Qu, Pratik Devasthale, Dennis Farrelly, Jeon Yoon T, Randolph P. Ponticiello, John R. Wetterau, Wei Wang, Wen-Pin Yang, Thomas Harrity, Aaron Tieman, Denis E. Ryono, Richard E. Gregg
Publikováno v:
Diabetes. 55:240-248
Muraglitazar, a novel dual (alpha/gamma) peroxisome proliferator-activated receptor (PPAR) activator, was investigated for its antidiabetic properties and its effects on metabolic abnormalities in genetically obese diabetic db/db mice. In db/db mice
Autor:
Denis E. Ryono, Chen Sean, Pratik Devasthale, Shu Y Chang, John R. Wetterau, W. Griffith Humphreys, Gary J. Grover, Dennis Farrelly, Jeon Yoon T, Fucheng Qu, Ramakrishna Seethala, Narayanan Hariharan, Wei Wang, Zhengping Ma, Scott A. Biller, Rajasree Golla, Lisa Moore, Arthur M. Doweyko, Michael Cap, Fred Selan, Jimmy Ren, Paul G. Sleph, Hao Zhang, Aaron Tieman, Vito G. Sasseville, Thomas Harrity, Gamini Chandrasena, Chunning Shao, Peter T. W. Cheng, Lin Cheng, Wei Sun
Publikováno v:
Journal of Medicinal Chemistry. 48:2248-2250
Muraglitazar/BMS-298585 (2) has been identified as a non-thiazolidinedione PPAR alpha/gamma dual agonist that shows potent activity in vitro at human PPARalpha (EC(50) = 320 nM) and PPARgamma(EC(50) = 110 nM). Compound 2 shows excellent efficacy for
Autor:
Thomas, Harrity, Dennis, Farrelly, Aaron, Tieman, Cuixia, Chu, Lori, Kunselman, Liqun, Gu, Randolph, Ponticiello, Michael, Cap, Fucheng, Qu, Chunning, Shao, Wei, Wang, Hao, Zhang, William, Fenderson, Sean, Chen, Pratik, Devasthale, Yoon, Jeon, Ramakrishna, Seethala, Wen-Pin, Yang, Jimmy, Ren, Min, Zhou, Denis, Ryono, Scott, Biller, Kasim A, Mookhtiar, John, Wetterau, Richard, Gregg, Peter T, Cheng, Narayanan, Hariharan
Publikováno v:
Diabetes. 55(1)
Muraglitazar, a novel dual (alpha/gamma) peroxisome proliferator-activated receptor (PPAR) activator, was investigated for its antidiabetic properties and its effects on metabolic abnormalities in genetically obese diabetic db/db mice. In db/db mice
Autor:
Karen Brown, Sergio A. Lira, Narayanan Hariharan, Jianming Ren, Kasim A. Mookhtiar, Aaron Tieman, Richard E. Gregg, Deborah Hagan, Dennis Farrelly
The importance of glucokinase (GK; EC 2.7.1.12 ) in glucose homeostasis has been demonstrated by the association of GK mutations with diabetes mellitus in humans and by alterations in glucose metabolism in transgenic and gene knockout mice. Liver GK
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::b8ff419851905f6892e2f9c7b601e8bb
https://europepmc.org/articles/PMC24467/
https://europepmc.org/articles/PMC24467/