Anti-helminthic Activity of Consolida orientalis (Gay) Schröd. on Caenorhabditis elegans Nematodes and Determination of Possible Active Ingredients

Autor: Hulya Ozpinar

Publikováno v: Turkish Journal of Agriculture: Food Science and Technology, Vol 9, Iss 8, Pp 1593-1598 (2021)

Helminthiasis is an important parasitic disease, many of which are zoonotic, particularly common in developing countries and, in countries with hot and humid climates. Intestinal parasites can cause significant manifestations at all levels of the gas

Externí odkaz: https://doaj.org/article/3073eedea8de4c588b3971bff8c29364

Microwave-assisted synthesis and pharmacological screening of some triazolothiadiazole derivatives

Autor: Ozge Gorgu, Engin Yıldırım, Yesim Ozkan, Bilge Cakır, Kevser Erol, Tijen Onkol

Publikováno v: Brazilian Journal of Pharmaceutical Sciences, Vol 56 (2020)

In this study, twenty-two new [1,2,4]triazolo[3,4-b][1,3,4]thiadiazoles (5a-n, 6a-h) were synthesized under microwave irradiation (MWI). The chemical structures of the compounds were elucidated by their IR, 1H-NMR, LC-MS, and elemental analysis. The

Externí odkaz: https://doaj.org/article/afb7435755f243e3ab2b76c40b5bde2c

Investigation of some 3-substituted-2(3H)-benzoxazolone derivatives against caspase-3 : A molecular docking study

Autor: null Emine Erdag

In the development of pharmacological probes, 2(3H)-benzoxazolones are viewed as privileged scaffolds. The functionalization of the nitrogen atom at the third position of the 2(3H)-benzoxazolone moiety is of importance because the electrical properti

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::052d6fe62af8e80cef219c468a338c6f

6-[(4-Chlorophenyl)(1H-1,2,4-triazol-1-yl)methyl]-3-methyl-2(3H)-benzoxazolone

Autor: Mariana S. Gerova, Yordanka B. Ivanova, Christo D. Chanev, Ognyan I. Petrov

Publikováno v: Molbank, Vol 2016, Iss 2, p M901 (2016)

A new hybrid molecule containing a triazole and a benzoxazolone ring was synthesized. The structure of 6-[(4-chlorophenyl)(1H-1,2,4-triazol-1-yl) methyl]-3-methyl-2(3H)-benzoxazolone was confirmed by IR, 1H-, 13C-NMR, MS and elemental analysis.

Externí odkaz: https://doaj.org/article/d092d39bd1ef4019a6a50278ec5b34af

Microwave-assisted synthesis and pharmacological screening of some triazolothiadiazole derivatives

Autor: Kevser Erol, Yeşim Özkan, Tijen Önkol, Bilge Çakir, Engin Yildirim, Ozge Gorgu

Publikováno v: Brazilian Journal of Pharmaceutical Sciences, Vol 56 (2020)
Brazilian Journal of Pharmaceutical Sciences, Volume: 56, Article number: e18111, Published: 16 MAR 2020
Brazilian Journal of Pharmaceutical Sciences; Vol. 56 (2020); e18111
Brazilian Journal of Pharmaceutical Sciences; v. 56 (2020); e18111
Brazilian Journal of Pharmaceutical Sciences
Universidade de São Paulo (USP)
instacron:USP

In this study, twenty-two new [1,2,4]triazolo[3,4-b][1,3,4]thiadiazoles (5a-n, 6a-h) were synthesized under microwave irradiation (MWI). The chemical structures of the compounds were elucidated by their IR, 1 H-NMR, LC-MS, and elemental analysis. The

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::b6cd1815c1ee68a851e07779b11b6232
http://www.scielo.br/scielo.php?script=sci_arttext&pid=S1984-82502020000100526&tlng=en