Zobrazeno 1 - 10
of 125
pro vyhledávání: '"δ receptor"'
Publikováno v:
Proceedings of the National Academy of Sciences of the United States of America, 1981 Oct 01. 78(10), 6181-6185.
Externí odkaz:
https://www.jstor.org/stable/11031
Akademický článek
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Akademický článek
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Autor:
Dietis, Nikolas, Niwa, H., Tose, R., McDonald, J., Ruggieri, V., Filaferro, M., Vitale, G., Micheli, L., Ghelardini, C., Salvadori, S., Calo, G., Guerrini, R., Rowbotham, D. J., Lambert, D. G.
Publikováno v:
British Journal of Pharmacology
Background and Purpose Targeting more than one opioid receptor type simultaneously may have analgesic advantages in reducing side-effects. We have evaluated the mixed μ opioid receptor agonist/ δ opioid receptor antagonist UFP-505 in vitro and in v
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::9ce6a1da77e7ae8279b1755238366f9a
http://hdl.handle.net/11577/3386314
http://hdl.handle.net/11577/3386314
Autor:
Kremer, Mélanie
La douleur neuropathique est due à une lésion ou une pathologie du système nerveux somatosensoriel. La prégabaline, un anticonvulsivant, et la duloxétine, un antidépresseur, sont des traitements de référence, efficaces chez un tiers des patie
Externí odkaz:
http://www.theses.fr/2016STRAJ033/document
Autor:
Nam Joo Hong, Dong Hee Kim
Publikováno v:
Bulletin of the Korean Chemical Society. 33:261-269
The cyclic dimers of enkephalin were isolated as minor components during the solution synthesis of the corresponding cyclic monomers. The ratio of cyclic dimer to monomer was approximately 1:4 from the percent of yields. In the receptor binding assay
Publikováno v:
Neurobiology of Disease, Vol 13, Iss 1, Pp 63-73 (2003)
We previously reported differential alterations of the mu, delta, and kappa opioid receptors following permanent middle cerebral artery occlusion. The present work studied the evolution of opioid receptor types following transient focal cerebral isch
Autor:
G. Weltrowska, Peter W. Schiller, N. N. Chung, T. M.-D. Nguyen, B. C. Wilkes, Katharine A. Carpenter, Carole Lemieux, Irena Berezowska, Ralf Schmidt
Publikováno v:
Journal of Receptors and Signal Transduction. 19:573-588
The development of novel delta opioid antagonists and delta opioid agonists structurally derived from the prototype delta antagonist TIPP (H-Tyr-Tic-Phe-Phe-OH), is reviewed. Both delta antagonists and delta agonists with extraordinary potency and un
Autor:
Ralf Schmidt, Nga N. Chung, Peter W. Schiller, Grazyna Weltrowska, Sébastien Dupuis, Carole Lemieux, Katharine A. Carpenter, Brian C. Wilkes, Irena Berezowska, Thi M.-D. Nguyen
Publikováno v:
Letters in Peptide Science. 5:209-214
Novel conformationally constrained opioid peptide analogs with δ antagonist, mixed μ agonist/δ antagonist or δ agonist properties were developed. TIP(P)-related δ antagonists showed unprecedented δ antagonist potency and δ receptor selectivity
Publikováno v:
Experimental and Therapeutic Medicine
Alpinetin is a natural flavonoid that protects cells against fatal injury in ischemia-reperfusion. δ receptor activation protects myocardial cells from trauma; however, the mechanism is unknown. The aim of this study was to explore the function of a