Zobrazeno 1 - 6
of 6
pro vyhledávání: '"Ágota Szájli"'
Autor:
Balázs Lendvai, Anna E. Káncz, Pál Tapolcsányi, Zoltán Béni, János Kóti, Marta Than, Éva Bozó, János Éles, István Greiner, Judit Laszy, Zsolt Némethy, Sándor Mahó, András Visegrády, Márton Vass, Gyula Bugovits, György Lévay, István Ledneczki, Anikó Pocsai, Balázs Krámos, Ágota Szájli, Mónika Vastag, Patrik Holm, Sándor Kolok, Eszter Gábor, Ottilia Balázs, Anita Horváth, József Nagy
Publikováno v:
European Journal of Medicinal Chemistry. 214:113189
The paper focuses on the scaffold hopping-based discovery and characterization of novel nicotinic alpha 7 receptor positive modulator (α7 nAChR PAM) ligands around the reference molecule (A-867744). First, substantial efforts were carried out to ass
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::a3ad9ffda37f8a3d089c88187d8a3c0f
https://doi.org/10.1016/j.ejmech.2021.113189
https://doi.org/10.1016/j.ejmech.2021.113189
Publikováno v:
The Journal of Organic Chemistry. 76:6048-6056
Ionic liquids 1-butyl-3-methylimidazolium hexafluorophosphate ([bmim](+)[PF(6)](-)) and 1-butyl-3-methylimidazolium tetrafluoroborate ([bmim](+)[BF(4)](-)) were found to promote an unusual Wagner-Meerwein rearrangement of steroidal 16α,17α-epoxides
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::bd52a11a5212bd4a9b7a5f22aa6e40c2
https://doi.org/10.1021/jo2006285
https://doi.org/10.1021/jo2006285
Autor:
Ágota Szájli, Zsófia Hoyk, Eszter Csakvari, Stephan Rühl, Andrea Gyenes, János Kóti, János Wölfling, Árpád Párducz, Roland Pfoh, Gábor Paragi
Publikováno v:
Steroids. 75:265-271
The naturally occurring steroid dehydroepiandrosterone (DHEA) is reported to reduce glial fibrillary acidic protein (GFAP) overexpression in a model of reactive gliosis due to its conversion to estradiol by the enzyme aromatase. In the present study
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::09898d767b180e0902640652e59a973a
https://doi.org/10.1016/j.steroids.2010.01.001
https://doi.org/10.1016/j.steroids.2010.01.001
Autor:
Ágota Szájli, János Wölfling
Publikováno v:
Monatshefte für Chemie - Chemical Monthly. 137:1431-1440
16-Ketene dithioacetal derivatives of 3β-hydroxy-13α-androst-5-en-17-one react with amidine, benzamidine, or guanidine to yield novel pyrimido-fused D-heteroannulated steroids. The reactions of 3β-hydroxy-16-hydroxymethylidene-13α-androst-5-en-17
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::3df75f71c5597d02405c9944ff93fa62
https://doi.org/10.1007/s00706-006-0544-7
https://doi.org/10.1007/s00706-006-0544-7
Publikováno v:
Monatshefte für Chemie - Chemical Monthly. 137:1099-1107
3β-Hydroxy-16,17-seco-13α-androsta-5,16-dien-17-al was obtained from 3β-acetoxyandrost-5-en-17-one in six steps with a Grob fragmentation as the key step. This seco-steroid, containing a formyl group and an unsaturated side-chain in a sterically f
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::6d1e1a223e7fd06bb9003c20ed1457d1
https://doi.org/10.1007/s00706-005-0500-y
https://doi.org/10.1007/s00706-005-0500-y
Autor:
Ágota Szájli, Gyula Schneider, Erzsébet Mernyák, George Falkay, Árpád Márki, János Wölfling, Renáta Minorics
Publikováno v:
Steroids. 71:141-153
The four possible isomers of 3-benzyloxy-16-hydroxymethylestra-1,3,5(10)-trien-17-ol (1a-4a) with proven configurations were converted into the corresponding 3-benzyloxy-16-bromomethylestra-1,3,5(10)-triene-3,17-diols (5e-8e). Depending on the reacti
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::21355b7bad99286781344c1a8497377c
https://doi.org/10.1016/j.steroids.2005.09.008
https://doi.org/10.1016/j.steroids.2005.09.008