Zobrazeno 1 - 6
of 6
pro vyhledávání: '"Kiyoshi Inoguchi"'
Autor:
Motonori Miyakawa, Noriko Yamamoto, Naoya Nagata, Kazuyuki Furuya, Kiyoshi Inoguchi, Seiji Amano, Hiroaki Nejishima
Publikováno v:
Bioorganic & Medicinal Chemistry Letters. 21:6310-6313
A rationally designed tetrahydroquinoline (1) for nonsteroidal selective androgen receptor modulators was modified for the exploration of promising compounds by Grieco three-component condensation using various dienophiles. Based on the in vitro effe
Autor:
Yasuo Yoneda, Mitsuo Hayashida, Shinji Tauchi, Akinori Aoyama, Tadashi Okuno, Nobuo Ishiyama, Kiyoshi Inoguchi, Mitsuo Mimura, Kiyoharu Ukai, Hirohide Ishige, Takeshi Kiyofuji
Publikováno v:
HETEROCYCLES. 67:561
The discovery and the SAR of acylproline derivatives as highly potent growth hormone secretagogues (GHSs) with good oral bioavailability are described. One representative compound, N-[3-(2,2-dimethylpropylamino)-2-hydroxypropyl]-2(R)-[l-(2,2-dimethyl
Publikováno v:
HETEROCYCLES. 56:257
The reaction of N-protected 3-pyrrolidone and 4-piperidone with N,N-dimethylformamide dimethyl acetal gave the dimethylaminomethylene ketones, which reacted with several types of hydrazines, amidines, and guanidine to afford the secondary amines havi
Publikováno v:
HETEROCYCLES. 31:1413
We prepared a modified DIOP analogue bearing bis(4-dimethylamino-3,5-dimethylphenyl)phosphino groups. Its rhodium complex was found to be a useful catalysts for asymmetric hydrogenation of dimethyl itaconate and itaconic acid derivatives bearing β-a
Autor:
Ryuichi Sakagami, Kazuo Ohta, Ryuichiro Tamada, Yoshio Hara, Kozo Jikuya, Tetsuo Taguchi, Kintomo Takakura, Satoru Kusama, Yasuo Koyama, Ryunosuke Kumashiro, Yukio Imamura, Yoshiyuki Koyama, Makoto Ogawa, Tatuo Saito, Osamu Takatani, Keiichi Maruyama, Noritsugu Umeda, Teruo Sakano, Minoru Murakami, Yukoh Inoue, Isao Nakao, Tadashi Kimura, Yosuke Nakano, Kenzo Okabayashi, Takeshi Tominaga, Nobuo Okazaki, Yasunobu Sakai, Kiyoshi Inoguchi, Akira Kubo, Ichiji Itoh, Osamu Nakajima, Jiro Tomiyama, Hisanobu Niitani, Takao Kanko, Yasuhiko Oh-hashi, Masakazu Yokoyama, Toru Ise, Jun-ichi Ishiwata
Publikováno v:
Japanese Journal of Clinical Oncology. 10:83-91
Autor:
Akira Wakui, Tetsuo Taguchi, Hisashi Majima, Tatsuo Saito, Shoji Suga, Ichiro Urushizaki, Kiyoji Kimura, Ota K, Hisanobu Niitani, Hidehito Ichihashi, Takao Hattori, Osahiko Abe, Kiyoshi Inoguchi, Ryuzo Ohno, Kazumasa Yamada, Hisashi Furue, Yozo Suzuoki
Publikováno v:
Cancer Chemotherapy and Pharmacology. 20:223-229
A phase I clinical and pharmacokinetic study of recombinant human tumor necrosis factor (rH-TNF) was conducted in a single dose schedule in 33 patients with advanced cancer. rH-TNF was given by i.v. infusion over 30 min with a starting dose of 1 x 10