Zobrazeno 1 - 8
of 8
pro vyhledávání: '"Pascale Coric"'
Autor:
Marie-Claude Fournie-Zaluski, Brigitte Barbe, Nathalie Rousselet, Pascale Coric, Jean-Baptiste Michel, Serge Turcaud, Isabelle Pham, Nathalie Jullian, Walter D. Gonzalez, Bernard P. Roques
Publikováno v:
Journal of Medicinal Chemistry
Journal of Medicinal Chemistry, 1994, 37 (8), pp.1070-1083. ⟨10.1021/jm00034a005⟩
Journal of Medicinal Chemistry, American Chemical Society, 1994, 37 (8), pp.1070-1083. ⟨10.1021/jm00034a005⟩
Journal of Medicinal Chemistry, 1994, 37 (8), pp.1070-1083. ⟨10.1021/jm00034a005⟩
Journal of Medicinal Chemistry, American Chemical Society, 1994, 37 (8), pp.1070-1083. ⟨10.1021/jm00034a005⟩
In the treatment of cardiovascular diseases, it could be of therapeutic interest to associate the hypotensive effects resulting from the inhibition of angiotensin II formation, ensured by endothelial angiotensin-converting enzyme (ACE), with the diur
Autor:
Bernard P. Roques, Evelyne Lucas, Florence Noble, Pascale Coric, Serge Turcaud, Luce Bruetschy, Marie Claude Fournie-Zaluski
Publikováno v:
Journal of Medicinal Chemistry
Journal of Medicinal Chemistry, American Chemical Society, 1992, 35 (7), pp.1259-1266. ⟨10.1021/jm00085a013⟩
Journal of Medicinal Chemistry, American Chemical Society, 1992, 35 (7), pp.1259-1266. ⟨10.1021/jm00085a013⟩
Derivatives of amino acids bearing various zinc-coordinating moieties (SH, COOH, CONHOH, and PO3H2) were synthesized and tested for their ability to inhibit aminopeptidase N (APN). Among them, beta-amino thiols were found to be the most efficient wit
Autor:
Pascal George, Aurélie Mothé, Sophie Danascimento, Huixiong Chen, Marie-Claude Fournie-Zaluski, Florence Noble, Hervé Meudal, Pascale Coric, Bernard P. Roques
Publikováno v:
Journal of Medicinal Chemistry
Journal of Medicinal Chemistry, American Chemical Society, 2000, 43 (7), pp.1398-408
Journal of Medicinal Chemistry, American Chemical Society, 2000, 43 (7), pp.1398-1408. ⟨10.1021/jm990483l⟩
HAL
Journal of Medicinal Chemistry, American Chemical Society, 2000, 43 (7), pp.1398-408
Journal of Medicinal Chemistry, American Chemical Society, 2000, 43 (7), pp.1398-1408. ⟨10.1021/jm990483l⟩
HAL
International audience; The development of dual inhibitors of the two zinc metallopeptidases, neprilysin (neutral endopeptidase) and aminopeptidase N involved in the inactivation of the opioid peptides, enkephalins, represents an attractive physiolog
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::0d955abead22b714e8d98f04de2a9de9
https://hal.archives-ouvertes.fr/hal-02122153
https://hal.archives-ouvertes.fr/hal-02122153
Autor:
Marie-Claude Fournie-Zaluski, Huixiong Chen, Bernard P. Roques, Pascale Coric, Florence Noble
Publikováno v:
Proceedings of the National Academy of Sciences of the United States of America
Proceedings of the National Academy of Sciences of the United States of America, National Academy of Sciences, 1998, 95 (20), pp.12028-12033. ⟨10.1073/pnas.95.20.12028⟩
Proceedings of the National Academy of Sciences of the United States of America, 1998, 95 (20), pp.12028-12033. ⟨10.1073/pnas.95.20.12028⟩
Proceedings of the National Academy of Sciences of the United States of America, National Academy of Sciences, 1998, 95 (20), pp.12028-12033. ⟨10.1073/pnas.95.20.12028⟩
Proceedings of the National Academy of Sciences of the United States of America, 1998, 95 (20), pp.12028-12033. ⟨10.1073/pnas.95.20.12028⟩
Inhibition of aminopeptidase N and neutral endopeptidase-24.11, two zinc metallopeptidases involved in the inactivation of the opioid peptides enkephalins, produces potent physiological analgesic responses, without major side-effects, in all animal m
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::ca64b162a2570e4d21ad4514343f807e
https://hal.archives-ouvertes.fr/hal-03456417
https://hal.archives-ouvertes.fr/hal-03456417
Autor:
Pascale Coric, Claire Smadja, Marie Claude Fournie-Zaluski, Rafael Maldonado, Bernard P. Roques, Fernando Ruiz
Publikováno v:
Psychopharmacology
Psychopharmacology, Springer Verlag, 1997, 132 (3), pp.227-236. ⟨10.1007/s002130050340⟩
Psychopharmacology, 1997, 132 (3), pp.227-236. ⟨10.1007/s002130050340⟩
Psychopharmacology, Springer Verlag, 1997, 132 (3), pp.227-236. ⟨10.1007/s002130050340⟩
Psychopharmacology, 1997, 132 (3), pp.227-236. ⟨10.1007/s002130050340⟩
Systemic administration of RB 101, a complete inhibitor of enkephalin catabolism, has been reported to induce antidepressant-like responses in mice which were potentiated by an ineffective dose of a CCK-B antagonist. The aim of this study was to inve
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::7bc70ac8cb27633c5c320417635120f7
https://hal.archives-ouvertes.fr/hal-02461428
https://hal.archives-ouvertes.fr/hal-02461428
Autor:
Pascale Coric, Claire Smadja, Rafael Maldonado, Olga Valverde, Marie-Claude Fournie-Zaluski, Serge Turcaud, Florence Noble, Bernard P. Roques
Publikováno v:
PAIN
PAIN, Elsevier, 1997, 73 (3), pp.383-391. ⟨10.1016/S0304-3959(97)00125-5⟩
Pain
Pain, 1997, 73 (3), pp.383-391. ⟨10.1016/S0304-3959(97)00125-5⟩
PAIN, Elsevier, 1997, 73 (3), pp.383-391. ⟨10.1016/S0304-3959(97)00125-5⟩
Pain
Pain, 1997, 73 (3), pp.383-391. ⟨10.1016/S0304-3959(97)00125-5⟩
RB 101 (N-((R,S)-2-benzyl-3[(S)(2-amino-4-methylthio)butyldithio]-1-oxopr opyl)-L-phenylalanine benzyl ester) is a full inhibitor of the enkephalin-catabolizing enzymes, which induces strong naloxone-reversible antinociceptive responses after i.v. or
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::d2d5feb7191881569d831fdffcd917bd
https://hal.archives-ouvertes.fr/hal-02461424
https://hal.archives-ouvertes.fr/hal-02461424
Autor:
Walter Gonzalez, Vincent Thery, Bernard P. Roques, Jean-Baptiste Michel, Marie-Claude Fournie-Zaluski, Hervé Meudal, Pascale Coric, Serge Turcaud
Publikováno v:
Journal of Medicinal Chemistry
Journal of Medicinal Chemistry, 1996, 39 (13), pp.2594-2608. ⟨10.1021/jm950783c⟩
Journal of Medicinal Chemistry, American Chemical Society, 1996, 39 (13), pp.2594-2608. ⟨10.1021/jm950783c⟩
Journal of Medicinal Chemistry, 1996, 39 (13), pp.2594-2608. ⟨10.1021/jm950783c⟩
Journal of Medicinal Chemistry, American Chemical Society, 1996, 39 (13), pp.2594-2608. ⟨10.1021/jm950783c⟩
International audience; Mercaptoacyl dipeptides, containing a glycine linked to a C-terminal 5-phenylproline, have been synthesized in order to obtain new highly efficient dual inhibitors of the two zinc metallopeptidases, neutral endopeptidase (NEP)
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::6845a5103c7d44a4522001abb6ba9396
https://doi.org/10.1021/jm950783c
https://doi.org/10.1021/jm950783c
Publikováno v:
European Journal of Pharmacology
European Journal of Pharmacology, Elsevier, 1992, 223 (1), pp.91-96. ⟨10.1016/0014-2999(92)90822-L⟩
European Journal of Pharmacology, Elsevier, 1992, 223 (1), pp.91-96. ⟨10.1016/0014-2999(92)90822-L⟩
Development of physical dependence is observed after treatment with opioid agonists, but not after chronic i.c.v. administration of mixed inhibitors of enkephalin-degrading enzymes. The aim of this study was to investigate further this promising resu
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::d8a3a5a71b288eb6c95b6c34d36ae280
https://hal.archives-ouvertes.fr/hal-02461500
https://hal.archives-ouvertes.fr/hal-02461500