Zobrazeno 1 - 1
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pro vyhledávání: '"Grasso, S."'
Autor:
Ettore Novellino, Silvana Grasso, Tanja Schirmeister, Andrea Pinto, Antonio Lavecchia, Maria Zappalà, Roberta Ettari, Carmen Cerchia, Nicola Micale, Valeria Troiano, Kety Scarbaci
Publikováno v:
European Journal of Medicinal Chemistry. 83:1-14
A new series of pseudopeptide boronate proteasome inhibitors (2–3) was developed, through optimization of our previously described analogs of bortezomib, bearing a bicyclic 1,6-naphthyridin-5(6H)-one scaffold as P3 fragment (1). The biological eval