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Autor:
Louis D. Trombetta, Yves Pommier, Aaditya Bhatt, Tanaji T. Talele, John M. Pascal, Junko Murai, Adel Chergui, Jamin D. Steffen, Maulik R. Patel, Frank R. Fronczek
Publikováno v:
Journal of Medicinal Chemistry
Novel substituted 2,3-dihydrobenzofuran-7-carboxamide (DHBF-7-carboxamide) and 2,3-dihydrobenzofuran-3(2H)-one-7-carboxamide (DHBF-3-one-7-carboxamide) derivatives were synthesized and evaluated as inhibitors of poly(ADP-ribose)polymerase-1 (PARP-1).