Zobrazeno 1 - 3
of 3
pro vyhledávání: '"59"'
Autor:
Crawford TD; Genentech, Inc. 1 DNA Way, South San Francisco, California 94080, United States., Romero FA; Genentech, Inc. 1 DNA Way, South San Francisco, California 94080, United States., Lai KW; Wuxi Apptec Co., Ltd. , 288 Fute Zhong Road, Waigaoqiao Free Trade Zone, Shanghai 200131, People's Republic of China., Tsui V; Genentech, Inc. 1 DNA Way, South San Francisco, California 94080, United States., Taylor AM; Constellation Pharmaceuticals, Inc. 215 First Street, Suite 200, Cambridge, Massachusetts 02142, United States., de Leon Boenig G; Genentech, Inc. 1 DNA Way, South San Francisco, California 94080, United States., Noland CL; Genentech, Inc. 1 DNA Way, South San Francisco, California 94080, United States., Murray J; Genentech, Inc. 1 DNA Way, South San Francisco, California 94080, United States., Ly J; Genentech, Inc. 1 DNA Way, South San Francisco, California 94080, United States., Choo EF; Genentech, Inc. 1 DNA Way, South San Francisco, California 94080, United States., Hunsaker TL; Genentech, Inc. 1 DNA Way, South San Francisco, California 94080, United States., Chan EW; Genentech, Inc. 1 DNA Way, South San Francisco, California 94080, United States., Merchant M; Genentech, Inc. 1 DNA Way, South San Francisco, California 94080, United States., Kharbanda S; Genentech, Inc. 1 DNA Way, South San Francisco, California 94080, United States., Gascoigne KE; Genentech, Inc. 1 DNA Way, South San Francisco, California 94080, United States., Kaufman S; Genentech, Inc. 1 DNA Way, South San Francisco, California 94080, United States., Beresini MH; Genentech, Inc. 1 DNA Way, South San Francisco, California 94080, United States., Liao J; Wuxi Apptec Co., Ltd. , 288 Fute Zhong Road, Waigaoqiao Free Trade Zone, Shanghai 200131, People's Republic of China., Liu W; Wuxi Apptec Co., Ltd. , 288 Fute Zhong Road, Waigaoqiao Free Trade Zone, Shanghai 200131, People's Republic of China., Chen KX; Wuxi Apptec Co., Ltd. , 288 Fute Zhong Road, Waigaoqiao Free Trade Zone, Shanghai 200131, People's Republic of China., Chen Z; Wuxi Apptec Co., Ltd. , 288 Fute Zhong Road, Waigaoqiao Free Trade Zone, Shanghai 200131, People's Republic of China., Conery AR; Constellation Pharmaceuticals, Inc. 215 First Street, Suite 200, Cambridge, Massachusetts 02142, United States., Côté A; Constellation Pharmaceuticals, Inc. 215 First Street, Suite 200, Cambridge, Massachusetts 02142, United States., Jayaram H; Constellation Pharmaceuticals, Inc. 215 First Street, Suite 200, Cambridge, Massachusetts 02142, United States., Jiang Y; Wuxi Apptec Co., Ltd. , 288 Fute Zhong Road, Waigaoqiao Free Trade Zone, Shanghai 200131, People's Republic of China., Kiefer JR; Genentech, Inc. 1 DNA Way, South San Francisco, California 94080, United States., Kleinheinz T; Genentech, Inc. 1 DNA Way, South San Francisco, California 94080, United States., Li Y; Wuxi Apptec Co., Ltd. , 288 Fute Zhong Road, Waigaoqiao Free Trade Zone, Shanghai 200131, People's Republic of China., Maher J; Genentech, Inc. 1 DNA Way, South San Francisco, California 94080, United States., Pardo E; Constellation Pharmaceuticals, Inc. 215 First Street, Suite 200, Cambridge, Massachusetts 02142, United States., Poy F; Constellation Pharmaceuticals, Inc. 215 First Street, Suite 200, Cambridge, Massachusetts 02142, United States., Spillane KL; Constellation Pharmaceuticals, Inc. 215 First Street, Suite 200, Cambridge, Massachusetts 02142, United States., Wang F; Wuxi Apptec Co., Ltd. , 288 Fute Zhong Road, Waigaoqiao Free Trade Zone, Shanghai 200131, People's Republic of China., Wang J; Wuxi Apptec Co., Ltd. , 288 Fute Zhong Road, Waigaoqiao Free Trade Zone, Shanghai 200131, People's Republic of China., Wei X; Wuxi Apptec Co., Ltd. , 288 Fute Zhong Road, Waigaoqiao Free Trade Zone, Shanghai 200131, People's Republic of China., Xu Z; Wuxi Apptec Co., Ltd. , 288 Fute Zhong Road, Waigaoqiao Free Trade Zone, Shanghai 200131, People's Republic of China., Xu Z; Wuxi Apptec Co., Ltd. , 288 Fute Zhong Road, Waigaoqiao Free Trade Zone, Shanghai 200131, People's Republic of China., Yen I; Genentech, Inc. 1 DNA Way, South San Francisco, California 94080, United States., Zawadzke L; Constellation Pharmaceuticals, Inc. 215 First Street, Suite 200, Cambridge, Massachusetts 02142, United States., Zhu X; Wuxi Apptec Co., Ltd. , 288 Fute Zhong Road, Waigaoqiao Free Trade Zone, Shanghai 200131, People's Republic of China., Bellon S; Constellation Pharmaceuticals, Inc. 215 First Street, Suite 200, Cambridge, Massachusetts 02142, United States., Cummings R; Constellation Pharmaceuticals, Inc. 215 First Street, Suite 200, Cambridge, Massachusetts 02142, United States., Cochran AG; Genentech, Inc. 1 DNA Way, South San Francisco, California 94080, United States., Albrecht BK; Constellation Pharmaceuticals, Inc. 215 First Street, Suite 200, Cambridge, Massachusetts 02142, United States., Magnuson S; Genentech, Inc. 1 DNA Way, South San Francisco, California 94080, United States.
Publikováno v:
Journal of medicinal chemistry [J Med Chem] 2016 Dec 08; Vol. 59 (23), pp. 10549-10563. Date of Electronic Publication: 2016 Sep 28.
Autor:
Traquandi G; Nerviano Medical Sciences Srl, Business Unit Oncology, Viale Pasteur 10, 20014 Nerviano, MI, Italy. gabriella.traquandi@nervianoms.com, Ciomei M, Ballinari D, Casale E, Colombo N, Croci V, Fiorentini F, Isacchi A, Longo A, Mercurio C, Panzeri A, Pastori W, Pevarello P, Volpi D, Roussel P, Vulpetti A, Brasca MG
Publikováno v:
Journal of medicinal chemistry [J Med Chem] 2010 Mar 11; Vol. 53 (5), pp. 2171-87.
Autor:
Jonathan Maher, F. Anthony Romero, Samir Kharbanda, Mark Merchant, Ivana Yen, Yingjie Li, Edna F. Choo, Jiangpeng Liao, Xiaocang Wei, Kwong Wah Lai, Karen E. Gascoigne, Richard D. Cummings, Hariharan Jayaram, Thomas Hunsaker, Steven F. Bellon, Jian Wang, Cameron L. Noland, Brian K. Albrecht, Ying Jiang, Jeremy Murray, Susan Kaufman, Kerry L. Spillane, Florence Poy, Zhaowu Xu, Fei Wang, James R. Kiefer, Laura Zawadzke, Zhongguo Chen, Alexander M. Taylor, Andrew R. Conery, Xiaoyu Zhu, Wenfeng Liu, Eneida Pardo, Alexandre Côté, Andrea G. Cochran, Vickie Tsui, Steven Magnuson, Terry Crawford, Maureen Beresini, Emily Chan, Kevin X. Chen, Gladys de Leon Boenig, Justin Ly, Tracy Kleinheinz, Zhongya Xu
Publikováno v:
Journal of medicinal chemistry. 59(23)
The single bromodomain of the closely related transcriptional regulators CBP/EP300 is a target of much recent interest in cancer and immune system regulation. A co-crystal structure of a ligand-efficient screening hit and the CBP bromodomain guided i