Zobrazeno 1 - 2
of 2
pro vyhledávání: '"59"'
Autor:
Alessia Salvador, Paola Barraja, Daniela Vedaldi, Gaetano Dattolo, Giampietro Viola, Alessandra Montalbano, Girolamo Cirrincione, Giuseppe Basso, Annamaria Martorana, Francesco Dall'Acqua, Patrizia Diana
Publikováno v:
Journal of medicinal chemistry. 51(8)
Isoindoloquinoxalines 4 and 5 were obtained by refluxing 2-(2'-aminoaryl)-1-cyanoisoindoles 3a- e in acetic or formic acid. All derivatives were screened by the National Cancer Institute (Bethesda, MD) for the in vitro one dose primary anticancer ass
Autor:
Madeleine Blanc, Luc Choisnard, Denis Wouessidjewe, Edwige Nicolle, Pierre-Alain Carrupt, Annabelle Gèze, Eva-Laure Matera, Ahcène Boumendjel, Charles Dumontet, Julien Boccard
Publikováno v:
Journal of Medicinal Chemistry, Vol. 51, No 7 (2008) pp. 2307-10
A series of 59 chalcones was prepared and evaluated for the antimitotic effect against K562 leukemia cells. The most active chalcones were evaluated for their antiproliferative activity against a panel of 11 human and murine cell cancer lines. We fou