Zobrazeno 1 - 1
of 1
pro vyhledávání: '"Ciomei M"'
Autor:
Arturo Galvani, Roberto Cairoli, Matteo G. Della Porta, Alessandro Di Sanzo, Cristina Davite, Roberta Bosotti, Erika Ravelli, Francesco Fiorentini, Lucia Zanetta, Elena Colajori, Elena Ardini, Antonella Isacchi, Marina Ciomei, Frank Xiaodong Gan, Federico Lussana, Rosalinda Gatto, Giuseppe Rossi, Romana Pulci, Andrea Lombardi Borgia, Alessandro Rambaldi
Publikováno v:
Blood. 134:3855-3855
Background: NMS-03592088 is a novel, potent inhibitor of the FLT3, CSF1R and KIT receptor tyrosine kinases (KD < 1 nM for all three targets). The compound demonstrated high preclinical efficacy following oral administration in all tested target-depen